Leveraging machine learning and the Free-Wilson approach in lead optimization: Efficient discovery of a new chemical class modulating the GABAA α5 receptor

Michael Bieler

Janus Larsen

Tino Dyhring

Thomas Jacobsen

Karin Nielsen

Heike Schauerte

Yunhai Cui

Stefan Peters

Niklas Heine

Christian Eickmeier

Roberto Arban

Florian Montel

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