From protein to candidate: Discovery of EPZ-5676, a potent and selective inhibitor of the histone methyltransferase DOT1L

Richard Chesworth

Edward Olhava

Kevin Kuntz

Aravind Basavapathruni

Christina Majer

Chris Sneeringer

Christina Allain

Alejandra Raimondi

Christine Klaus

Margaret Porter Scott

Carly Therkelsen

Scott Daigle

Roy Pollock

Victoria Richon

Robert Copeland

P. Boriack-sjodin

Lei Jin

Nigel Waters

Lee Arnold

Michael Patane

Paul Pearson

Joelle Sacks

Mikel Moyer