Discovery and structure-based optimization of substituted 4-hydroxy-5,6-dihydropyran/dihydropyridin-2-ones as potent inhibitors of human lactate dehydrogenase A

Binqing Wei

Kirk Robarge

Sharada Labadie

Aihe Zhou

Benjamin Fauber

Peter Dragovich

Zhenting Gao

Charles Ding

Tommy Lai

Laura Corson

Anna Hitz

Mark Ultsch

Charles Eigenbrot

Ivana Yen

Laurent Salphati

Thomas O'brien

Hans E Purkey

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