Discovery of a novel class of potent, selective, and orally bioavailable histone methyltransferase Enhancer of Zeste Homolog 2 (EZH2) inhibitors and the identification of development candidate PF-06821497

Pei-pei Kung

Simon Bergqvist

Patrick Bingham

John Braganza

Alexei Brooun

Michael Collins

Wade Diehl

Ya-li Deng

Dinh Dac

Connie Fan

Valeria Fantin

Hovhannes Gukasyan

Wenyue Hu

Buwen Huang

Robert Kania

Wei Liu

Susan Kephart

Manfred Kraus

Cody Krivacic

Robert Kumpf

Gary Li

Karen Maegley

Indrawan J McAlpine

Lisa Nguyen

Sacha Ninkovic

Martha A Ornelas

Dan Richter

Eugene Rui

Michael Ryskin

Stephanie A Scales

Jillian Spangler

Al Stewart

Scott Sutton

John Tatlock

Cheng-chung Tsao

Dominique Verhelle

Fen Wang

Hui Wang

Peter Wells

Martin Wythes

Shinji Yamazaki

Brian Yip

Xiu Yu

Luke Zehnder

Wei-guo Zhang

Peter Zhu

Jinjiang Zhu

Robert Rollins

Shikhar Sharma

Martin Edwards

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