High-throughput experimentation (HTE) plays a pivotal role in drug discovery and development, and as the synthesis of medicinal chemistry targets and libraries expand beyond amidations and SnAr reactions to more challenging chemo- and bio-catalyzed transformations, balancing cost, speed, and quality become paramount. Herein, we present ongoing efforts to accelerate early portfolio utilizing HTE detailing successes, failures, and culminating in program-enabling strategies impacting medicinal chemistry and chemical research and development.

Program enabling strategies utilizing HTE

Fall 2022 abstracts, posters, and presentations will launch in mid-September.

ACS Fall 2022

The official archive and repository for all ACS Meetings & Expositions abstracts and select posters or presentations.